SCHEMBL14420183

SCHEMBL14420183

COc1ccc2c(c1)/C(=C/CCN1CCC(c3ccc(O)cc3)CC1)c1cccnc1CO2

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.47
CHRM2 P08172 1/20 0.47
CCR5 P51681 1/20 0.47
DRD2 P14416 4/20 0.38
DRD4 P21917 2/20 0.38
CARM1 Q86X55 2/20 0.37
TBXA2R P21731 2/20 0.36
HTR1A P08908 1/20 0.36
HTR2A P28223 1/20 0.36
DRD3 P35462 1/20 0.36
APP P05067 1/20 0.35
HRH1 P35367 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7211997 0.93 CCR1 (0.47) CCR1CHRM2CCR5DRD2DRD4
SCHEMBL7212000 0.93 CCR1 (0.47) CCR1CHRM2CCR5DRD2DRD4
SCHEMBL7212913 0.92 CCR1 (0.54) CCR1CHRM2CCR5DRD2DRD4
SCHEMBL7212910 0.92 CCR1 (0.54) CCR1CHRM2CCR5DRD2DRD4
SCHEMBL10287856 0.90 CCR1 (0.46) CCR1CHRM2CCR5DRD2DRD4
SCHEMBL7207268 0.88 CCR1 (0.49) CCR1CHRM2CCR5TBXA2RHRH1
SCHEMBL7207266 0.88 CCR1 (0.49) CCR1CHRM2CCR5TBXA2RHRH1
SCHEMBL13824388 0.88 CCR1 (0.46) CCR1CHRM2CCR5DRD2DRD4
SCHEMBL10287855 0.88 CCR1 (0.46) CCR1CHRM2CCR5DRD2DRD4
SCHEMBL14419953 0.86 CCR1 (0.56) CCR1CHRM2CCR5DRD2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7271176-B2 Chemokine receptor antagonists and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-09-18 US disclosed