SCHEMBL14422752

SCHEMBL14422752

N#Cc1ccc(Nc2nnc3ccc(NC4CC4)nn23)cc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 8/20 0.48
MALT1 Q9UDY8 9/20 0.43
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
CDK2 P24941 2/20 0.40
CCNK O75909 1/20 0.40
CCNA2 P20248 1/20 0.40
CDK12 Q9NYV4 1/20 0.40
CCNE1 P24864 1/20 0.40
FLT3 P36888 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14422755 0.86 PIM1 (0.54) PIM1MALT1CDK2FLT3
SCHEMBL14422761 0.84 PIM1 (0.65) PIM1MALT1CDK2FLT3CYP3A4
SCHEMBL14422795 0.84 PIM1 (0.64) PIM1MALT1CDK2FLT3CYP3A4
SCHEMBL14422734 0.81 ABCG2 (0.47) FLT3
SCHEMBL14422765 0.81 PIM1 (0.67) PIM1MALT1CDK2FLT3CYP3A4
SCHEMBL14422680 0.81 PIM1 (0.71) PIM1MALT1CDK2FLT3
SCHEMBL14422759 0.75 PIM1 (0.65) PIM1MALT1CDK2FLT3
SCHEMBL14422748 0.74 KDM4E (0.43) CDK2FLT3CYP2C9CYP2C19
SCHEMBL14422768 0.73 MALT1 (0.72) PIM1MALT1CDK2FLT3KCNH2
SCHEMBL14422769 0.73 PIM1 (0.67) PIM1MALT1CDK2FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7268136-B2 Compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-09-11 US disclosed