SCHEMBL14423907

SCHEMBL14423907

CC(C)N(C)CCn1nc(-c2cccc(Br)c2)c2cnccc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.34
ALDH1A1 P00352 3/20 0.33
NPSR1 Q6W5P4 3/20 0.33
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GAA P10253 1/20 0.33
KCNA5 P22460 2/20 0.33
LMNA P02545 4/20 0.33
CNR1 P21554 3/20 0.33
GPR55 Q9Y2T6 3/20 0.33
CNR2 P34972 2/20 0.33
HTT P42858 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
PKM P14618 1/20 0.33
CYP2C19 P33261 1/20 0.33
PPARG P37231 1/20 0.33
NR2E3 Q9Y5X4 1/20 0.33
NCOR2 Q9Y618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9304627 0.89 CYP2D6 (0.41) CYP2D6ALDH1A1NPSR1KDM4EMEN1
Hydrochloric Acid SCHEMBL8142868 0.88 CYP2D6 (0.40) CYP2D6ALDH1A1NPSR1KDM4EMEN1
SCHEMBL9303541 0.85 CYP2D6 (0.47) CYP2D6ALDH1A1KDM4EGAACYP1A2
Hydrochloric Acid SCHEMBL8127101 0.83 CYP2D6 (0.46) CYP2D6ALDH1A1KDM4EGAACYP1A2
Hydrochloric Acid SCHEMBL9263878 0.83 CYP2D6 (0.46) CYP2D6ALDH1A1KDM4EGAACYP1A2
SCHEMBL9305917 0.81 HRH1 (0.38) ALDH1A1NPSR1KDM4EMEN1KMT2A
SCHEMBL5359047 0.81 KDM4E (0.38) CYP2D6ALDH1A1NPSR1KDM4EMEN1
SCHEMBL9303549 0.79 KDM4E (0.39) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL9304434 0.76 CYP2D6 (0.42) CYP2D6ALDH1A1NPSR1CYP1A2CYP2C9
SCHEMBL9305128 0.76 CYP2D6 (0.50) CYP2D6ALDH1A1KDM4EKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7253165-B2 Benzisoxazolyl-, pyridoisoxazolyl-and benzthienyl-phenoxy derivatives useful as D4 antagonists AVENTIS PHARMACEUTICALS INC. (US) 2007-08-07 US disclosed