SCHEMBL9305917

SCHEMBL9305917

NCCn1nc(-c2cccc(Br)c2)c2cnccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
KDM4E B2RXH2 2/20 0.36
HSD17B10 Q99714 2/20 0.36
TSHR P16473 1/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
KCNH2 Q12809 2/20 0.35
ALDH1A1 P00352 3/20 0.35
GAA P10253 1/20 0.35
CYP19A1 P11511 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303549 0.93 KDM4E (0.39) HRH1HRH4KDM4EHSD17B10TSHR
SCHEMBL8137072 0.86 ALDH1A1 (0.39) KDM4EHSD17B10TSHRMAPTALDH1A1
SCHEMBL9306122 0.86 HSD17B10 (0.47) KDM4EHSD17B10TSHRKMT2ALMNA
SCHEMBL9304627 0.85 CYP2D6 (0.41) KDM4EHSD17B10TSHRMEN1KMT2A
SCHEMBL5359047 0.85 KDM4E (0.38) KDM4EHSD17B10TSHRMEN1KMT2A
Hydrochloric Acid SCHEMBL8134231 0.84 HSD17B10 (0.46) KDM4EHSD17B10TSHRKMT2ALMNA
Hydrochloric Acid SCHEMBL8142868 0.84 CYP2D6 (0.40) KDM4EMEN1KMT2ALMNAMAPT
SCHEMBL9303541 0.83 CYP2D6 (0.47) KDM4EHSD17B10TSHRKCNH2ALDH1A1
SCHEMBL9258008 0.83 NAMPT (0.39) KDM4EHSD17B10TSHRMAPTMERTK
Hydrochloric Acid SCHEMBL8127101 0.81 CYP2D6 (0.46) KDM4EHSD17B10TSHRKCNH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296491-A Pyrazolo[4,3-c]pyridines and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-22 US claimed