SCHEMBL14435008

SCHEMBL14435008

CC1CCC(C(=O)Nc2ccc3c(c2)CCNCC3)N1C(=O)Nc1ccc(Br)cc1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MELK Q14680 3/20 0.55
KDM4E B2RXH2 1/20 0.40
SLC2A1 P11166 1/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
NAMPT P43490 1/20 0.38
HPGD P15428 1/20 0.37
FLT3 P36888 1/20 0.37
MAPT P10636 1/20 0.37
FPR3 P25089 1/20 0.37
FPR2 P25090 1/20 0.37
CFD P00746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12371477 0.89 NPC1 (0.43) MELKKDM4EKMT2AMEN1NPC1
SCHEMBL14435010 0.79 MELK (0.51) MELKKDM4ESLC2A1KMT2AMEN1
SCHEMBL14434240 0.79 MELK (0.51) MELKKDM4ESLC2A1KMT2AMEN1
SCHEMBL12371463 0.79 MELK (0.51) MELKKDM4ESLC2A1KMT2AMEN1
SCHEMBL14435007 0.77 MELK (0.49) MELKKDM4ESLC2A1KMT2AMEN1
SCHEMBL14435246 0.75 MELK (0.47) MELKKDM4ESLC2A1KMT2AMEN1
SCHEMBL12371429 0.71 KDM4E (0.50) MELKKDM4EKMT2AMEN1NPC1
SCHEMBL12101393 0.71 NPC1 (0.42) KMT2AMEN1NPC1RAB9AHCRTR1
SCHEMBL14434686 0.69 SLC2A1 (0.51) MELKSLC2A1CFD
SCHEMBL12371426 0.69 MEN1 (0.53) MELKKDM4EKMT2AMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007093595-A1 SUBSTITUTED PROLINAMIDES, THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-08-23 WO disclosed