SCHEMBL14435443

SCHEMBL14435443

Cc1c(O)nc(C2CC2)nc1CO

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 9/20 0.42
CHRM3 P20309 9/20 0.36
PDE4A P27815 7/20 0.36
PDE4B Q07343 7/20 0.36
PDE4C Q08493 7/20 0.36
PDE4D Q08499 7/20 0.36
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TKT P29401 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL276474 0.82 PDE10A (0.54) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL14435742 0.77 PDE10A (0.39) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL13769264 0.76 PDE10A (0.48) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL11185504 0.74 PDE10A (0.42) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL4428463 0.74 PDE10A (0.45) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL4419009 0.74 PDE10A (0.45) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL909717 0.69 CHRM3 (0.43) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL4424922 0.68 PDE10A (0.39) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL4429098 0.68 PDE10A (0.39) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL717059 0.67 TSHR (0.38) PDE10AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007089031-A1 PIPERIDINE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-09 WO disclosed