SCHEMBL14459752

SCHEMBL14459752

[O-][n+]1c(Cl)c(Cl)cc(Cl)c1Cl

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.37
MAPK1 P28482 1/20 0.35
AHR P35869 1/20 0.35
TSHR P16473 3/20 0.32
HPGD P15428 2/20 0.32
HSD17B10 Q99714 2/20 0.32
CASP1 P29466 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11822900 0.65
SCHEMBL348913 0.64 AHR (0.67) CYP3A4MAPK1AHRTSHRHPGD
SCHEMBL8773848 0.64
SCHEMBL30461566 0.62 NMT1 (0.35)
SCHEMBL10040909 0.62
SCHEMBL25219379 0.62 NMT1 (0.35)
SCHEMBL5843888 0.62 TSHR (0.39) TSHR
SCHEMBL8773850 0.61 CYP3A4 (0.32) CYP3A4MAPK1AHR
SCHEMBL4300949 0.57 CYP3A4 (0.41) CYP3A4MAPK1AHRTSHRHPGD
SCHEMBL877968 0.57

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7262210-B2 Fluorinated pyridine N-oxide thrombin modulators and process for N-oxidation of nitrogen containing heteroaryls JANSSEN PHARMACEUTICA N.V. (BE) 2007-08-28 US disclosed