SCHEMBL14459986

SCHEMBL14459986

CCCCN1CCN(Cc2c(F)cccc2Cl)CC1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A13 Q16696 1/20 0.61
ALDH1A1 P00352 2/20 0.60
TDP1 Q9NUW8 2/20 0.60
ALOX15 P16050 1/20 0.60
DRD2 P14416 2/20 0.58
DRD3 P35462 2/20 0.58
CACNA1G O43497 5/20 0.58
KDM4E B2RXH2 3/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
TSHR P16473 2/20 0.54
POLB P06746 1/20 0.54
SIGMAR1 Q99720 2/20 0.53
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
LMNA P02545 2/20 0.49
HTR1A P08908 1/20 0.49
DRD4 P21917 1/20 0.49
HTR2A P28223 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12732277 0.96 CYP2A13 (0.59) CYP2A13ALDH1A1TDP1ALOX15DRD2
SCHEMBL14608742 0.91 CYP2A13 (0.64) CYP2A13ALDH1A1TDP1ALOX15DRD2
SCHEMBL656160 0.87 CYP2A13 (0.62) CYP2A13ALDH1A1TDP1ALOX15CACNA1G
SCHEMBL12709637 0.85 CYP2A13 (0.57) CYP2A13ALDH1A1TDP1ALOX15CACNA1G
SCHEMBL19998608 0.80 CYP2A13 (0.61) CYP2A13ALDH1A1TDP1ALOX15CACNA1G
SCHEMBL18939695 0.80 DRD2 (0.64) CYP2A13ALDH1A1TDP1ALOX15DRD2
SCHEMBL11938897 0.77 DRD2 (0.48) CYP2A13ALDH1A1DRD2DRD3KDM4E
SCHEMBL209940 0.76 CYP2A13 (0.68) CYP2A13ALDH1A1TDP1ALOX15CACNA1G
SCHEMBL16256924 0.76 KDM4E (0.68) CYP2A13ALDH1A1DRD2DRD3KDM4E
SCHEMBL4107051 0.76 CYP2A13 (1.00) CYP2A13ALDH1A1TDP1ALOX15CACNA1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1813616-A2 Pyrazoloquinolines with immunomodulating activity Active Biotech AB (SE) 2007-08-01 EP disclosed
EP-1562944-B1 PYRAZOLOQUINOLINES WITH IMMUNOMODULATING ACTIVITY ACTIVE BIOTECH AB (SE) 2007-02-14 EP disclosed