SCHEMBL14465623

SCHEMBL14465623

CCCn1cncc1CCN

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
MTOR P42345 1/20 0.35
HRH4 Q9H3N8 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
CYP11B1 P15538 10/20 0.34
CYP11B2 P19099 10/20 0.34
ADORA2A P29274 2/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16803390 0.86 CYP11B1 (0.37) CYP11B1CYP11B2ADORA2AADORA2BADORA1
SCHEMBL1785054 0.85 KCNH2 (0.40) CYP2C9TSHRCYP2C19MTORHRH4
SCHEMBL12064369 0.83 CYP11B1 (0.41) CYP2C9CYP2C19HRH3CYP11B1CYP11B2
SCHEMBL15996487 0.80 ADORA2A (0.33) CYP2C9CYP2C19CYP11B1CYP11B2ADORA2A
SCHEMBL12056295 0.79 IDO1 (0.39) CYP11B1CYP11B2
SCHEMBL8830161 0.79 CYP11B1 (0.39) CYP11B1CYP11B2
SCHEMBL21558721 0.77 KCNH2 (0.34) CYP11B1CYP11B2ADORA2AADORA2BADORA1
SCHEMBL5391398 0.77 CYP11B1 (0.45) CYP11B1CYP11B2ADORA2AADORA2BADORA1
SCHEMBL20439593 0.77 KCNH2 (0.34) ADORA2B
SCHEMBL14415973 0.76 CYP11B1 (0.33) CYP2C9TSHRCYP2C19MTORHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007084498-A1 PIPERAZINE DERIVATIVES AS FARNESYL PROTEIN TRANSFERASE INHIBITORS SCHERING CORPORATION (US) 2007-07-26 WO disclosed