SCHEMBL14465752

SCHEMBL14465752

CCc1cnc(N2CCN(S(=O)(=O)C[C@]34CC[C@](C)(CC3=O)C4(C)C)CC2)nc1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 8/20 0.49
L3MBTL1 Q9Y468 1/20 0.43
KDM4E B2RXH2 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
MMP13 P45452 9/20 0.39
MMP14 P50281 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5316606 0.78 CXCR3 (0.80) CXCR3L3MBTL1
SCHEMBL14466693 0.66 CXCR3 (0.70) CXCR3
SCHEMBL17414136 0.64 CYP1A2 (0.31)
SCHEMBL14465702 0.64
SCHEMBL17637714 0.64 CYP1A2 (0.31)
SCHEMBL3651006 0.63 OGA (0.46) KDM4ENPC1RAB9A
SCHEMBL14238181 0.62 HDAC3 (0.49) KDM4ENPC1RAB9A
SCHEMBL12503186 0.62 OGA (0.47) KDM4ENPC1RAB9A
SCHEMBL12525139 0.62 OGA (0.47) KDM4ENPC1RAB9A
SCHEMBL12913814 0.62 HDAC3 (0.65) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007076318-A2 CAMPHOR-DERIVED CXCR3 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed