SCHEMBL1446964

SCHEMBL1446964

O=C(O)C1CC[C@H](C(=O)c2ccc(-c3cnc(Nc4cccc(Cl)c4)nc3)cc2)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.50
HDAC1 Q13547 2/20 0.50
HDAC2 Q92769 2/20 0.50
HDAC6 Q9UBN7 2/20 0.50
DGAT1 O75907 2/20 0.49
CAMK2D Q13557 1/20 0.47
EGFR P00533 5/20 0.46
BTK Q06187 4/20 0.45
CSNK2A2 P19784 1/20 0.44
CSNK2B P67870 1/20 0.44
CSNK2A1 P68400 1/20 0.44
MGLL Q99685 1/20 0.42
CSF1R P07333 1/20 0.41
GFRA3 O60609 1/20 0.41
RET P07949 1/20 0.41
CNR2 P34972 3/20 0.40
SCN9A Q15858 1/20 0.40
BRAF P15056 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4D Q08499 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1448287 0.89 DGAT1 (0.50) HDAC3HDAC1HDAC2HDAC6DGAT1
SCHEMBL180651 0.86 DGAT1 (0.68) HDAC3HDAC1HDAC2HDAC6DGAT1
SCHEMBL1447834 0.86 DGAT1 (0.68) HDAC3HDAC1HDAC2HDAC6DGAT1
SCHEMBL180870 0.77 DGAT1 (0.61) DGAT1CAMK2DMGLLCSF1R
SCHEMBL180650 0.74 DGAT1 (0.69) DGAT1CSNK2A2CSNK2BCSNK2A1
SCHEMBL180868 0.70 DGAT1 (0.60) DGAT1
SCHEMBL180531 0.70 DGAT1 (0.62) DGAT1
SCHEMBL180931 0.70 DGAT1 (0.60) DGAT1
SCHEMBL180532 0.70 DGAT1 (0.62) DGAT1
SCHEMBL180533 0.70 DGAT1 (0.62) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2301923-A1 New compounds Novartis AG (CH) 2011-03-30 EP disclosed