SCHEMBL14495342

SCHEMBL14495342

Nc1ncnc(O)c1NCC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.44
GRIN3B O60391 1/20 0.44
GRIN1 Q05586 1/20 0.44
GRIN2A Q12879 1/20 0.44
GRIN2B Q13224 1/20 0.44
GRIN2C Q14957 1/20 0.44
GRIN3A Q8TCU5 1/20 0.44
PLAU P00749 2/20 0.38
KDM4E B2RXH2 2/20 0.35
MAP4K4 O95819 1/20 0.34
EGLN1 Q9GZT9 2/20 0.33
EGFR P00533 1/20 0.33
CHEK1 O14757 1/20 0.33
XDH P47989 1/20 0.33
MET P08581 1/20 0.32
APEX1 P27695 1/20 0.32
MAPT P10636 1/20 0.32
HIF1A Q16665 1/20 0.32
SLC22A6 Q4U2R8 1/20 0.32
SLC22A8 Q8TCC7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11035691 0.70 DNM2 (0.40) ALDH1A1
SCHEMBL28888193 0.67 KDR (0.35) MAP4K4XDHMETMAPTALDH1A1
SCHEMBL12590748 0.65 AKR1B1 (0.40) KDM4EAPEX1MAPTHIF1AGABRP
SCHEMBL16597183 0.64 KDM4E (0.41) KDM4EEGFRXDHAPEX1GABRP
Hydrochloric Acid SCHEMBL3760711 0.64 PI4KA (0.35) KDM4EMAP4K4CHEK1XDHMET
SCHEMBL1482970 0.62 GRIN2D (0.44) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9204756 0.62 GRIN2D (1.00) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL18773443 0.62 MAP4K4 (0.47) KDM4EMAP4K4EGFRMAPTTP53
SCHEMBL558620 0.61
SCHEMBL29439831 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007064553-A2 THIAZOLE DERIVATIVES AS CXCR3 RECEPTOR MODULATORS MERCK & CO., INC. (US) 2007-06-07 WO disclosed