SCHEMBL14501784

SCHEMBL14501784

CN(C)c1ccc2c(c1)CCC(CN1CCCC1)C2

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.46
HTR1A P08908 3/20 0.45
OPRM1 P35372 1/20 0.44
OPRL1 P41146 1/20 0.44
KDM2B Q8NHM5 1/20 0.41
HRH3 Q9Y5N1 3/20 0.40
MCHR1 Q99705 2/20 0.40
ALDH1A1 P00352 1/20 0.40
OPRD1 P41143 1/20 0.40
HRH1 P35367 1/20 0.39
BACE1 P56817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5383054 0.79 SIGMAR1 (0.48) SIGMAR1HTR1AOPRM1OPRL1HRH3
SCHEMBL5904201 0.79 CYP19A1 (0.53) SIGMAR1HTR1AOPRM1OPRL1HRH3
SCHEMBL5904101 0.78 SIGMAR1 (0.71) SIGMAR1HTR1AOPRM1OPRL1HRH3
SCHEMBL4621851 0.78 CYP19A1 (0.52) SIGMAR1HTR1AOPRM1OPRL1HRH3
SCHEMBL5582559 0.78 SIGMAR1 (0.47) SIGMAR1HTR1AOPRM1OPRL1HRH3
Bromide SCHEMBL5904342 0.78 CYP19A1 (0.52) SIGMAR1HTR1AOPRM1OPRL1HRH3
Hydrochloric Acid SCHEMBL4622114 0.77 CYP19A1 (0.51) SIGMAR1HTR1AOPRM1OPRL1HRH3
Hydrochloric Acid SCHEMBL4622628 0.76 SIGMAR1 (0.68) SIGMAR1HTR1AHRH3MCHR1HRH1
SCHEMBL14454746 0.76 SIGMAR1 (0.70) SIGMAR1HTR1AOPRM1OPRL1HRH3
Hydrochloric Acid SCHEMBL5904107 0.76 HRH3 (0.55) SIGMAR1HTR1AHRH3HRH1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7220777-B2 Lactam derivatives as antagonists for human 11cby receptors SMITHKLINE BEECHAM P.L.C. (GB) 2007-05-22 US disclosed
US-7220777-B2 Lactam derivatives as antagonists for human 11cby receptors SMITHKLINE BEECHAM P.L.C. (GB) 2007-05-22 US disclosed