SCHEMBL14517848

SCHEMBL14517848

CCCn1c(=O)c2[nH]c(-c3ccn[nH]3)nc2n(CCC)c1=O

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 12/20 0.64
ADORA2A P29274 6/20 0.64
KDM4E B2RXH2 1/20 0.64
MEN1 O00255 1/20 0.64
ALDH1A1 P00352 1/20 0.64
CYP1A2 P05177 1/20 0.64
CYP3A4 P08684 1/20 0.64
CYP2C9 P11712 1/20 0.64
CYP2C19 P33261 1/20 0.64
KMT2A Q03164 1/20 0.64
HSD17B10 Q99714 1/20 0.64
ADORA1 P30542 2/20 0.61
ADORA3 P0DMS8 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25090453 0.79 ADORA2B (0.60) ADORA2BADORA2AKDM4EALDH1A1CYP1A2
SCHEMBL661108 0.78 ADORA2B (1.00) ADORA2BADORA2AKDM4EMEN1ALDH1A1
SCHEMBL14564546 0.77 ADORA2B (0.79) ADORA2BADORA2AKDM4EMEN1ALDH1A1
SCHEMBL7318202 0.76 ADORA2B (1.00) ADORA2BADORA2AKDM4EMEN1ALDH1A1
SCHEMBL1948455 0.76 ADORA2B (1.00) ADORA2BADORA2AKDM4EMEN1ALDH1A1
SCHEMBL242345 0.75 ADORA2B (1.00) ADORA2BADORA2AKDM4EMEN1ALDH1A1
SCHEMBL8872400 0.75 ADORA2B (0.69) ADORA2BADORA2AKDM4EMEN1ALDH1A1
SCHEMBL7313540 0.74 ADORA2B (0.78) ADORA2BADORA2AKDM4EMEN1ALDH1A1
SCHEMBL10675027 0.74 ADORA2B (0.70) ADORA2BADORA2AKDM4EMEN1ALDH1A1
SCHEMBL10674822 0.74 ADORA2B (0.70) ADORA2BADORA2AKDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7205403-B2 8-Heteroaryl xanthine adenosine A2B receptor antagonists KING PHARMACEUTICALS RESEARCH AND DEVELOPMENT, INC. (US) 2007-04-17 US disclosed
US-7205403-B2 8-Heteroaryl xanthine adenosine A2B receptor antagonists KING PHARMACEUTICALS RESEARCH AND DEVELOPMENT, INC. (US) 2007-04-17 US disclosed