SCHEMBL14525367

SCHEMBL14525367

COC(=O)c1cn(C[C@H]2CN(c3ccc(C4=CC[S+]([O-])CC4)c(F)c3)C(=O)O2)nn1

nearest known ligand 0.63

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAOA P21397 18/20 0.63
KCNH2 Q12809 1/20 0.44
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5657103 1.00 MAOA (0.63) MAOAKCNH2CYP3A4CYP2D6
SCHEMBL14525376 0.90 MAOA (0.57) MAOAKCNH2CYP3A4CYP2D6
SCHEMBL5654671 0.87 MAOA (0.56) MAOAKCNH2
SCHEMBL14525377 0.87 MAOA (0.56) MAOAKCNH2
SCHEMBL4014908 0.87 MAOA (0.71) MAOAKCNH2CYP3A4CYP2D6
SCHEMBL13939803 0.87 MAOA (0.71) MAOAKCNH2CYP3A4CYP2D6
SCHEMBL5657622 0.86 MAOA (0.72) MAOAKCNH2CYP3A4CYP2D6
SCHEMBL14525371 0.86 MAOA (0.72) MAOAKCNH2CYP3A4CYP2D6
SCHEMBL5656542 0.84 MAOA (0.61) MAOAKCNH2CYP3A4CYP2D6
SCHEMBL5658912 0.84 MAOA (0.58) MAOAKCNH2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7199143-B2 Chemical compounds ASTRAZENECA AB (SE) 2007-04-03 US disclosed