SCHEMBL14529005

SCHEMBL14529005

NC(=O)Cc1nc2c(C(F)(F)F)cccc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGES O14684 3/20 0.51
PARP1 P09874 3/20 0.49
CHEK1 O14757 1/20 0.48
CCR2 P41597 6/20 0.44
MAOB P27338 1/20 0.43
CACNA1H O95180 4/20 0.43
CACNA1B Q00975 1/20 0.42
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1359506 0.87 CCR2 (0.47) PTGESPARP1CHEK1CCR2CACNA1H
SCHEMBL3367539 0.86 CCR2 (0.46) PTGESPARP1CHEK1CCR2CACNA1H
Lithium Ion SCHEMBL3367542 0.85 CHEK1 (0.44) PTGESPARP1CHEK1CCR2CACNA1H
SCHEMBL3372968 0.82 CHEK1 (0.70) PTGESPARP1CHEK1CCR2KDM4E
SCHEMBL16176683 0.78 CACNA1B (0.54) PTGESCCR2CACNA1HCACNA1BKDM4E
SCHEMBL4064263 0.78 CACNA1H (0.43) PARP1CACNA1HCACNA1B
SCHEMBL14529004 0.78 MAOB (0.43) PTGESPARP1MAOBCACNA1HKDM4E
SCHEMBL1360362 0.75 CCR2 (0.52) PTGESPARP1CCR2CACNA1H
SCHEMBL21200019 0.74 KDM4E (0.52) PARP1KDM4EHPGD
SCHEMBL19494475 0.73 CACNA1H (0.46) PTGESPARP1CCR2CACNA1HCACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007053498-A1 COMPOUNDS USEFUL AS ANTAGONISTS OF CCR2 MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-05-10 WO disclosed
WO-2007053499-A2 COMPOUNDS USEFUL AS ANTAGONISTS OF CCR2 MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-05-10 WO disclosed