SCHEMBL14529239

SCHEMBL14529239

Cc1ccc(-n2nc(C(=O)N3CCC[C@@H]3CF)cc2-c2ccccn2)nn1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 5/20 0.44
SCD5 Q86SK9 1/20 0.39
HCRTR1 O43613 6/20 0.36
HCRTR2 O43614 3/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
DAGLB Q8NCG7 1/20 0.35
DAGLA Q9Y4D2 1/20 0.35
ADORA2A P29274 2/20 0.34
ADORA1 P30542 2/20 0.34
GRM5 P41594 1/20 0.34
ABL1 P00519 1/20 0.34
RIN1 Q13671 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5270446 0.90 NTRK1 (0.42) NTRK1SCD5HCRTR1HCRTR2NPC1
SCHEMBL5271916 0.90 NTRK1 (0.42) NTRK1SCD5HCRTR1HCRTR2NPC1
SCHEMBL14529197 0.88 KDM4E (0.44) NTRK1SCD5HCRTR1GRM5
SCHEMBL13213189 0.82 NTRK1 (0.41) NTRK1SCD5
SCHEMBL14529778 0.81 ADORA2A (0.43) NTRK1ADORA2A
SCHEMBL5268570 0.81 ADORA2A (0.44) NTRK1SCD5HCRTR1HCRTR2NPC1
SCHEMBL5267292 0.81 KDM5A (0.34) NTRK1SCD5HCRTR1NPC1RAB9A
SCHEMBL14529496 0.80 ALDH1A1 (0.45) NTRK1SCD5NPC1RAB9A
SCHEMBL14529775 0.80 KCNJ6 (0.36) NTRK1HCRTR1HCRTR2
SCHEMBL5269213 0.79 GRM5 (0.35) NTRK1SCD5HCRTR1HCRTR2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1785418-A1 PYRAZOLE DERIVATIVE DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2007-05-16 EP disclosed