SCHEMBL14540932

SCHEMBL14540932

COCCOc1cc2nccc(Oc3ccc(N)c(Cl)c3)c2cc1C(=O)NOC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 1/20 0.51
KDR P35968 18/20 0.47
AURKB Q96GD4 6/20 0.47
AURKA O14965 6/20 0.47
TEK Q02763 6/20 0.47
MET P08581 5/20 0.47
PDGFRA P16234 4/20 0.47
FLT1 P17948 3/20 0.47
RET P07949 3/20 0.47
PDGFRB P09619 2/20 0.47
KIT P10721 2/20 0.47
FGFR1 P11362 2/20 0.47
FLT4 P35916 2/20 0.47
RIPK2 O43353 1/20 0.47
ERN1 O75460 1/20 0.47
STK10 O94804 1/20 0.47
MAP3K6 O95382 1/20 0.47
ABL1 P00519 1/20 0.47
ESR1 P03372 1/20 0.47
ADORA3 P0DMS8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22505666 0.93 KDR (0.52) AXLKDRAURKBAURKATEK
SCHEMBL1892397 0.91 AXL (0.51) AXLKDRAURKBAURKATEK
SCHEMBL14540914 0.91 KDR (0.58) AXLKDRAURKBAURKATEK
SCHEMBL5364065 0.90 AXL (0.50) AXLKDRAURKBAURKATEK
SCHEMBL22505715 0.90 AXL (0.59) AXLKDRAURKBAURKATEK
SCHEMBL14540583 0.90 KDR (0.54) AXLKDRAURKBAURKATEK
SCHEMBL14540940 0.88 KDR (0.52) AXLKDRAURKBAURKATEK
SCHEMBL14540522 0.87 KDR (0.47) KDRAURKBAURKATEKMET
SCHEMBL1892843 0.87 RET (0.51) AXLKDRAURKBAURKATEK
SCHEMBL14540588 0.86 PDGFRA (0.48) AXLKDRAURKBAURKATEK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1777218-A1 Process for the preparation of 4-phenoxy quinoline derivatives Eisai R&D Management Co., Ltd. (JP) 2007-04-25 EP disclosed