SCHEMBL14540969

SCHEMBL14540969

C=CC(O)(c1ccc(C(=O)N(C)CCc2ccccc2)cc1)C(F)(F)F

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 5/20 0.72
ESRRG P62508 1/20 0.50
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
GRIA2 P42262 1/20 0.46
TGM2 P21980 1/20 0.44
NR1H3 Q13133 2/20 0.44
NR1H2 P55055 1/20 0.44
MCHR1 Q99705 1/20 0.43
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
TACR1 P25103 1/20 0.41
CDK4 P11802 1/20 0.41
CCND1 P24385 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4987436 0.84 MLYCD (1.00) MLYCDESRRGNR1H3NR1H2
SCHEMBL13431498 0.83 MLYCD (0.79) MLYCDESRRGMEN1KMT2ACYP2C9
SCHEMBL12133560 0.76 MLYCD (0.72) MLYCDESRRGMEN1KMT2AMCHR1
SCHEMBL257847 0.74 MLYCD (0.69) MLYCDESRRGMEN1KMT2AMCHR1
SCHEMBL13181408 0.73 MLYCD (0.64) MLYCDMEN1KMT2AROCK2ROCK1
SCHEMBL27891608 0.71 MLYCD (0.65) MLYCDESRRGMEN1KMT2ACYP2C9
SCHEMBL2945131 0.71 MLYCD (1.00) MLYCDMEN1KMT2ANR1H3NR1H2
SCHEMBL177498 0.71 MLYCD (0.64) MLYCDESRRGCYP2C9CYP2C19GRIA2
SCHEMBL3230674 0.70 MLYCD (0.78) MLYCDMEN1KMT2ANR1H3
SCHEMBL6631811 0.70 MLYCD (0.60) MLYCDESRRGKMT2AMCHR1ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1353662-B1 METHODS FOR THE TREATMENT OF DISEASES USING MALONYL-COA DECARBOX YLASE INHIBITORS CHUGAI PHARMACEUTICAL CO LTD (JP) 2007-04-18 EP disclosed