SCHEMBL145453

SCHEMBL145453

O=S(=O)(OCC(F)F)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.36
CA1 P00915 2/20 0.34
CA9 Q16790 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3521831 0.85 CA2 (0.36) CA2CA1CA9
SCHEMBL16115817 0.81 CA2 (0.34) CA2CA1CA9
SCHEMBL28673552 0.81 CA2 (0.34) CA2CA1
SCHEMBL18392909 0.81
SCHEMBL17629788 0.81 CA2 (0.37) CA2CA1
SCHEMBL19713240 0.79 CA2 (0.33) CA2CA1
SCHEMBL18762503 0.78 CA2 (0.35) CA2CA1CA9
SCHEMBL20267825 0.78 CA2 (0.35) CA2CA1CA9
SCHEMBL271903 0.78 CA2 (0.35) CA2CA1CA9
SCHEMBL780303 0.78 CA2 (0.35) CA2CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2614 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250161911-A1 POLYMERS FOR THE REMOVAL OF PFAS FROM AQUEOUS COMPOSITIONS, AND METHODS OF MAKING AND USING THE SAME GULF COAST ENVIRONMENTAL SYSTEMS LLC (DBA CONIFER SYSTEMS) 2025-05-22 US claimed
WO-2025106778-A1 POLYMERS FOR THE REMOVAL OF PFAS FROM AQUEOUS COMPOSITIONS, AND METHODS OF MAKING AND USING THE SAME LUTUM TECHNOLOGY, LLC (US) 2025-05-22 WO claimed
CN-118356775-A Novel fluorine functionalized alcohol amine-based absorbent for capturing sulfur dioxide in mixed gas, preparation method and application 大连理工大学 2024-07-19 CN claimed
CN-101611026-A Preparation method of (3R,4R) -N- (4-chlorphenyl) -1- (2, 2-difluoroethyl) -N' - [ 2-fluoro-4- (2-oxo-1 (2H) -pyridyl) phenyl ] -3, 4-pyrrolidine dicarboxamide HOFFMANN LA ROCHE (CH) 2009-12-23 CN claimed
EP-2097401-A1 PROCESSES FOR THE PREPARATION OF (3R, 4R) -N- (4 -CHLOROPHENYL) -1- (2, 2-DIFLUOROETHYL) -N' - [2-FLUORO-4- (2-OXO-1 (2H) -PYRIDINYL) PHENYL]-3, 4-PYRROLIDINEDICARBOXAMIDE F. Hoffmann-Roche AG (CH) 2009-09-09 EP claimed
US-20080214826-A1 PROCESSES FOR THE MANUFACTURE OF A PYRROLIDINE-3,4-DICARBOXAMIDE DERIVATIVE HOFFMANN-LA ROCHE, INC. 2008-09-04 US claimed
WO-2008077797-A1 PROCESSES FOR THE PREPARATION OF (3R, 4R) -N- (4 -CHLOROPHENYL) -1- (2, 2-DIFLUOROETHYL) -N' - [2-FLUORO-4- (2-OXO-1 (2H) -PYRIDINYL) PHENYL] -3, 4-PYRROLIDINEDICARBOXAMIDE F. HOFFMANN-LA ROCHE AG (CH) 2008-07-03 WO claimed
EP-4746963-A1 MACROCYCLES FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. Hoffmann-La Roche AG (CH) 2026-05-27 EP disclosed
WO-2026107418-A1 N-(4-(1H-BENZO[D[IMIDAZOL-6-YL)-PYRIDIN-2-YL)BENZAMIDE DERIVATIVES AS CAMK2 INHIBITORS FOR THE TREATMENT OF HEART FAILURE BRISTOL-MYERS SQUIBB COMPANY (US) 2026-05-21 WO disclosed
WO-2026103793-A1 TRICYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, AND USE THEREOF 上海翰森生物医药科技有限公司 2026-05-21 WO disclosed
WO-2026107424-A1 N-(4-(IMIDAZO[4,5-B]PYRIDIN-5-YL)-2-PYRIDYL)BENZAMIDE DERIVATIVES AS CAMK2 INHIBITORS FOR THE TREATMENT OF HEART FAILURE BRISTOL-MYERS SQUIBB COMPANY (US) 2026-05-21 WO disclosed
EP-4744661-A2 NOVEL PYRIMIDIN-2-YL SULFONAMIDE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2026-05-20 EP disclosed
EP-4743455-A1 SARM1 INHIBITORS F. Hoffmann-La Roche AG (CH) 2026-05-20 EP disclosed
US-6218364-B1 FOR THERAPY OF ASTHMA MERRELL PHARMACEUTICALS, INC. 2001-04-17 US disclosed
EP-1084137-A1 PEPTIDE INHIBITORS OF HEPATITIS C VIRUS NS3 PROTEASE ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2001-03-21 EP disclosed
WO-1999064442-A1 PEPTIDE INHIBITORS OF HEPATITIS C VIRUS NS3 PROTEASE ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P ANGELETTI S.P.A. (IT) 1999-12-16 WO disclosed
US-5750089-A Halogenated neuroprobe for mapping monoamine reuptake sites NEURO IMAGING TECHNOLOGIES, LLC (US) 1998-05-12 US disclosed
EP-0831941-A1 IODINATED NEUROPROBES FOR MAPPING MONOAMINE REUPTAKE SITES Research Biochemicals, Limited Paternership, doing business as Research biochemicals International (US) 1998-04-01 EP disclosed
US-5698179-A Iodinated neuroprobe for mapping monoamine reuptake sites NEURO IMAGING TECHNOLOGIES, LLC (US) 1997-12-16 US disclosed
WO-1996039198-A1 IODINATED NEUROPROBES FOR MAPPING MONOAMINE REUPTAKE SITES RESEARCH BIOCHEMICALS, LIMITED PARTNERSHIP, doing business as RESEARCH BIOCHEMICALS INTERNATIONAL, A MASSACHUSETTS LIMITED PARTNERSHIP, WHOSE SOLE GENERAL PARTNER IS RBI MANAGEMENT, INC. (US) 1996-12-12 WO disclosed