SCHEMBL145524

SCHEMBL145524

CCCNC(N)=S

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28115548 0.97
Methane SCHEMBL27965354 0.97
SCHEMBL144837 0.83
SCHEMBL28919 0.81
Pyrimidine SCHEMBL27529476 0.81 QPCT (0.37)
Pyridine SCHEMBL28880004 0.81 KMT2A (0.41)
SCHEMBL15344088 0.81 ALDH1A1 (0.48)
SCHEMBL15999308 0.80
SCHEMBL5570327 0.79 EPHX1 (0.54)
SCHEMBL7269038 0.79 EPHX1 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 633 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4590782-A1 GAS-PHASE COMPOSITION FOR INHIBITING CORROSION EXPOSED TO CONDENSED WATER Arkema France (FR) 2025-07-30 EP claimed
EP-3884921-B1 DENTAL POLYMERIZABLE COMPOSITION G C DENTAL IND CORP (JP) 2025-07-02 EP claimed
EP-3884922-B1 DENTAL POLYMERIZABLE COMPOSITION G C DENTAL IND CORP (JP) 2025-06-18 EP claimed
CN-119798537-A Biosensor, biosensor outer film, and preparation method and application of biosensor outer film 上海微创生命科技有限公司 2025-04-11 CN claimed
CN-119307989-A Electrolyte additive, electrolyte, copper foil, preparation method and application of electrolyte additive and copper foil 江西理工大学 2025-01-14 CN claimed
CN-119243226-A Two-dimensional molybdenum-based nano-sheet catalyst and preparation method and application thereof 重庆理工大学 2025-01-03 CN claimed
CN-118910406-A Method for enhancing bioleaching of chalcopyrite 中国科学院过程工程研究所 2024-11-08 CN claimed
CN-113906321-B Polarizing plate, method for manufacturing same, and image display device 住友化学株式会社 2024-10-15 CN claimed
EP-4441164-A1 FOAMING COMPOSITION COMPATIBLE WITH STEEL FOR THE ASSISTED RECOVERY OF HYDROCARBONS ARKEMA FRANCE (FR) 2024-10-09 EP claimed
WO-2024062191-A1 GAS-PHASE COMPOSITION FOR INHIBITING CORROSION EXPOSED TO CONDENSED WATER ARKEMA FRANCE (FR) 2024-03-28 WO claimed
EP-0752986-B1 N-HETEROCYCLYL SULPHONAMIDE DERIVATIVES AND THEIR USE AS ENDOTHELIN ANTAGONISTS ZENECA LTD (GB) 1999-05-19 EP claimed
US-5861401-A TREATMENT OF CONGESTIVE HEART FAILURE ZENECA LIMITED (GB) 1999-01-19 US claimed
EP-0832082-A1 N-HETEROARYL-PYRIDINESULFONAMIDE DERIVATIVES AND THEIR USE AS ENDOTHELIN ANTAGONISTS ZENECA LIMITED (GB) 1998-04-01 EP claimed
JP-H09510987-A 1997-11-04 JP claimed
US-5641793-A POSSESS ENDOTHELIN RECEPTOR ANTAGONIST ACTIVITY; USEFUL IN TREATMENT OF HYPERTENSION, CARDIAC OR CEREBRAL CIRCULATORY DISEASE AND RENAL DISEASE ZENECA LIMITED (GB) 1997-06-24 US claimed
EP-0752986-A1 N-HETEROCYCLYL SULPHONAMIDE DERIVATIVES AND THEIR USE AS ENDOTHELIN ANTAGONISTS ZENECA LIMITED (GB) 1997-01-15 EP claimed
WO-1996040681-A1 N-HETEROARYL-PYRIDINESULFONAMIDE DERIVATIVES AND THEIR USE AS ENDOTHELIN ANTAGONISTS ZENECA LIMITED (GB) 1996-12-19 WO claimed
EP-0682016-A1 Pyridine derivatives ZENECA LIMITED (GB) 1995-11-15 EP claimed
WO-1995026957-A1 N-HETEROCYCLYL SULPHONAMIDE DERIVATIVES AND THEIR USE AS ENDOTHELIN ANTAGONISTS ZENECA LIMITED (GB) 1995-10-12 WO claimed
US-4627968-A Synthesis of crystalline aluminosilicate with alkylurea or alkylthiourea ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1986-12-09 US claimed