SCHEMBL14554158

SCHEMBL14554158

CCC(C)(C)c1ccc2c(CC#N)c[nH]c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 3/20 0.49
MCL1 Q07820 1/20 0.38
HTR1D P28221 5/20 0.38
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36
CASP3 P42574 1/20 0.36
RAB9A P51151 1/20 0.36
ATM Q13315 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
TBXAS1 P24557 1/20 0.36
GPR84 Q9NQS5 2/20 0.36
HTR2A P28223 3/20 0.35
HTR1A P08908 2/20 0.35
HTR1B P28222 1/20 0.35
BCHE P06276 1/20 0.34
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8957520 0.87 CSNK2A1 (0.53) CSNK2A1HTR1DTBXAS1GPR84HTR2A
SCHEMBL6029337 0.81 CSNK2A1 (0.53) CSNK2A1TBXAS1GPR84
SCHEMBL13262495 0.80 MCL1 (0.48) MCL1HTR1DNPC1LMNAMAPK1
SCHEMBL11924849 0.77 CSNK2A1 (0.54) CSNK2A1HTR1DNPC1GPR84HTR2A
SCHEMBL18708142 0.76 CSNK2A1 (0.57) CSNK2A1GPR84HTR2AHTR2CHTR2B
SCHEMBL15074715 0.76 HTR2A (0.59) CSNK2A1HTR1DGPR84HTR2AHTR2C
SCHEMBL9001726 0.76 HTR1D (0.40) HTR1DNPC1HTR2AHTR1AHTR1B
SCHEMBL9006989 0.75 CFTR (0.38) MCL1HTR1DNPC1LMNAMAPK1
SCHEMBL273402 0.73 CSNK2A1 (0.57) CSNK2A1HTR1DGPR84HTR2AHTR1B
SCHEMBL29354243 0.73 CSNK2A1 (0.77) CSNK2A1GPR84HTR2AHTR1ABCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130011923-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-01-10 US disclosed