SCHEMBL14558181

SCHEMBL14558181

CN(C)c1cccc(Nc2cc(-c3ccccc3N)ncn2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 7/20 0.52
CYP2D6 P10635 6/20 0.52
CYP2C19 P33261 4/20 0.52
CLK4 Q9HAZ1 4/20 0.52
ALDH1A1 P00352 4/20 0.52
CYP3A4 P08684 3/20 0.52
MAPK1 P28482 3/20 0.52
TSHR P16473 1/20 0.52
LMNA P02545 2/20 0.52
EGFR P00533 1/20 0.49
CCNT1 O60563 8/20 0.47
CDK9 P50750 8/20 0.47
MAP4K4 O95819 2/20 0.46
CDK1 P06493 2/20 0.46
CDK4 P11802 2/20 0.46
CCNB1 P14635 2/20 0.46
CCND1 P24385 2/20 0.46
ABL2 P42684 2/20 0.46
GSK3A P49840 2/20 0.46
CDK7 P50613 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14558177 0.85 EGFR (0.47) CYP1A2CYP2D6CYP2C19CLK4ALDH1A1
SCHEMBL374166 0.82 EGFR (0.61) CYP1A2CYP2D6CYP2C19CLK4ALDH1A1
SCHEMBL4104463 0.79 CCNT1 (0.62) CYP1A2CYP2D6CYP2C19CLK4ALDH1A1
SCHEMBL4108904 0.78 CCNT1 (0.54) CYP1A2CYP2D6CYP2C19CLK4ALDH1A1
SCHEMBL14558179 0.77 CCNT1 (0.49) CYP1A2CYP2D6CYP2C19CLK4ALDH1A1
SCHEMBL374904 0.76 TNNI3K (0.57) EGFRMEN1KMT2AKDM1ANPC1
SCHEMBL27637021 0.76 CYP1A2 (0.59) CYP1A2CYP2D6CYP2C19CLK4ALDH1A1
SCHEMBL27700538 0.75 EGFR (0.54) CYP1A2CYP2D6CYP2C19CLK4ALDH1A1
SCHEMBL14558182 0.75 NPC1 (0.71) CYP1A2CYP2D6CYP2C19CLK4ALDH1A1
SCHEMBL4109262 0.71 CYP1A2 (0.53) CYP1A2CYP2D6CYP2C19CLK4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189729-B2 Methods and compositions as protein kinase inhibitors IRM LLC (BM) 2007-03-13 US disclosed
US-7189729-B2 Methods and compositions as protein kinase inhibitors IRM LLC (BM) 2007-03-13 US disclosed