SCHEMBL27700538

SCHEMBL27700538

CN(C)c1cccc(Nc2cc(N)ncn2)c1.N=C=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.54
NPC1 O15118 2/20 0.43
CDK1 P06493 1/20 0.43
CCNB1 P14635 1/20 0.43
CCNA2 P20248 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
CDK5 Q00535 1/20 0.43
CDK5R1 Q15078 1/20 0.43
TNNI3K Q59H18 6/20 0.41
KDM1A O60341 1/20 0.41
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
JAK3 P52333 1/20 0.39
NOS1 P29475 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
RAB9A P51151 1/20 0.39
SCN9A Q15858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL374166 0.92 EGFR (0.61) EGFRNPC1CDK1CCNB1CCNA2
SCHEMBL374904 0.78 TNNI3K (0.57) EGFRNPC1TNNI3KKDM1AMEN1
SCHEMBL14558182 0.77 NPC1 (0.71) EGFRNPC1TNNI3KKDM1AMEN1
SCHEMBL14558181 0.75 CYP1A2 (0.52) EGFRNPC1CDK1CCNB1CCNA2
SCHEMBL8798667 0.73 EGFR (0.61) EGFRCDK1CCNB1CCNA2CCNE1
SCHEMBL12517456 0.72 TNNI3K (0.81) EGFRTNNI3K
SCHEMBL4108904 0.72 CCNT1 (0.54) EGFRMEN1KMT2AUSP2ALDH1A1
SCHEMBL374636 0.72 CYP2D6 (0.51) EGFRNPC1CDK1CCNB1CCNA2
SCHEMBL14558177 0.71 EGFR (0.47) EGFRCDK1CCNB1CCNA2CDK2
SCHEMBL3431925 0.70 CDK1 (0.60) EGFRNPC1CDK1CCNB1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101035769-A Pyrimidine urea derivatives as kinase inhibitors NOVARTIS AG (CH) 2007-09-12 CN disclosed