SCHEMBL14559503

SCHEMBL14559503

NCC(=O)OCC1CC(c2ccc(-c3ccc(N4C[C@H](Cn5ccnn5)OC4=O)cc3F)cn2)=NO1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAOA P21397 17/20 0.62
CYP3A4 P08684 4/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4758912 1.00 MAOA (0.62) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL14559464 0.95 MAOA (0.61) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL4758755 0.92 MAOA (0.60) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL4758751 0.92 MAOA (0.60) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL6071030 0.92 MAOA (0.60) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL14559468 0.92 MAOA (0.65) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL14559474 0.92 MAOA (0.68) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL5365406 0.92 MAOA (0.58) MAOACYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL4701430 0.92 MAOA (0.62) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL4702593 0.92 MAOA (0.62) MAOACYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7192974-B2 Hydroxymethyl substituted dihydroisoxazole derivatives useful as antibiotic agents ASTRAZENECA AB (SE) 2007-03-20 US disclosed
US-7192974-B2 Hydroxymethyl substituted dihydroisoxazole derivatives useful as antibiotic agents ASTRAZENECA AB (SE) 2007-03-20 US disclosed