SCHEMBL14565670

SCHEMBL14565670

N[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCCC[C@@H]1NC(=O)c1ccc2ccccc2n1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SSTR3 P32745 1/20 0.51
ALDH1A1 P00352 2/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
TACR1 P25103 2/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNA7 P36544 1/20 0.42
CHRNA4 P43681 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14565672 0.90 SSTR3 (0.47) SSTR3ALDH1A1GAAMAPTTACR1
SCHEMBL14565669 0.89 SSTR3 (0.49) SSTR3TACR1
SCHEMBL5258116 0.86 SSTR3 (0.49) SSTR3TACR1CHRNB2CHRNA7CHRNA4
SCHEMBL5256700 0.81 SSTR3 (0.58) SSTR3ALDH1A1GAAMAPTMEN1
SCHEMBL14565583 0.81 SSTR3 (0.58) SSTR3ALDH1A1GAAMAPTMEN1
SCHEMBL5255157 0.81 SSTR3 (0.58) SSTR3ALDH1A1GAAMAPTMEN1
SCHEMBL5257922 0.78 SSTR3 (0.47) SSTR3ALDH1A1GAAMAPTMEN1
SCHEMBL5254842 0.78 SSTR3 (0.47) SSTR3ALDH1A1GAAMAPTMEN1
SCHEMBL6840775 0.78 SSTR3 (0.47) SSTR3ALDH1A1GAAMAPTMEN1
SCHEMBL5255112 0.76 SSTR3 (0.52) SSTR3ALDH1A1GAAMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453801-B1 SUBSTITUTED 2-AMINO-CYCLOALKANECARBOXAMIDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed