SCHEMBL6840775

SCHEMBL6840775

N#C[C@@H](NC(=O)[C@@H]1CCCCC1NC(=O)c1ccc2ccccc2n1)C1CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR3 P32745 1/20 0.47
SCN9A Q15858 4/20 0.42
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
RAB9A P51151 3/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
CNR2 P34972 2/20 0.39
HTT P42858 1/20 0.39
MAPT P10636 3/20 0.39
GAA P10253 2/20 0.39
MAPK1 P28482 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5254842 1.00 SSTR3 (0.47) SSTR3SCN9AALDH1A1MEN1KMT2A
SCHEMBL5257922 1.00 SSTR3 (0.47) SSTR3SCN9AALDH1A1MEN1KMT2A
SCHEMBL6839364 0.87 SMN1; SMN2 (0.41) RAB9ASMN1; SMN2MAPTKDM4ENPC1
SCHEMBL5256198 0.87 SMN1; SMN2 (0.41) RAB9ASMN1; SMN2MAPTKDM4ENPC1
SCHEMBL5258116 0.83 SSTR3 (0.49) SSTR3
SCHEMBL5340986 0.82 SSTR3 (0.46) SSTR3SCN9AALDH1A1MEN1KMT2A
SCHEMBL5340990 0.82 SSTR3 (0.46) SSTR3SCN9AALDH1A1MEN1KMT2A
SCHEMBL5257713 0.82 HPGDS (0.46) PDE3BPDE3A
SCHEMBL6838493 0.82 HPGDS (0.46) PDE3BPDE3A
SCHEMBL5255112 0.81 SSTR3 (0.52) SSTR3SCN9AALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6759428-B2 SUCH AS N-((1,2)-2-(((CYANO(CYCLOPROPYL)METHYL)AMINO)CARBONYL) CYCLOHEXYL)-1H-INDOLE-2-CARBOXAMIDE; CATHEPSIN K INHIBITORS ROCHE PALO ALTO LLC 2004-07-06 US disclosed