SCHEMBL14587205

SCHEMBL14587205

O=C(c1cn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)nn1)c1[nH]ncc1-c1ccccc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 2/20 0.44
TACR1 P25103 1/20 0.41
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
PTGES O14684 1/20 0.39
ALOX5 P09917 1/20 0.39
EPHB4 P54760 2/20 0.39
GPBAR1 Q8TDU6 7/20 0.38
EPAS1 Q99814 1/20 0.38
TEK Q02763 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
ROCK2 O75116 2/20 0.35
PIM1 P11309 2/20 0.35
GSK3B P49841 2/20 0.35
AURKB Q96GD4 2/20 0.35
PLK4 O00444 1/20 0.35
AURKA O14965 1/20 0.35
CHUK O15111 1/20 0.35
MAPK13 O15264 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4638586 0.83 TACR1 (0.42) TACR1GPBAR1EPAS1
SCHEMBL4637956 0.80 ALDH1A1 (0.46) TACR1GPBAR1EPAS1ALDH1A1PIM1
SCHEMBL14144832 0.76 TACR1 (0.37) TACR1GPBAR1EPAS1ALDH1A1LMNA
SCHEMBL4707969 0.72 CDC7 (0.42) TACR1ALDH1A1ROCK2PIM1GSK3B
SCHEMBL4638855 0.71 EPAS1 (0.50) TACR1HSP90AA1HSP90AB1GPBAR1EPAS1
SCHEMBL5795073 0.71 HSP90AA1 (0.53) TGM2HSP90AA1HSP90AB1ALDH1A1LMNA
SCHEMBL4639409 0.68 TACR1 (0.39) TACR1GPBAR1EPAS1ALDH1A1
SCHEMBL2378228 0.68 P2RX1 (0.53) TGM2EPAS1ALDH1A1LMNA
SCHEMBL5797524 0.68 ALDH1A1 (0.50) TACR1GPBAR1ALDH1A1
SCHEMBL5797317 0.67 HSP90AA1 (0.58) TGM2HSP90AA1HSP90AB1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7179804-B2 Tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 2007-02-20 US disclosed
US-7179804-B2 Tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 2007-02-20 US disclosed