SCHEMBL14587739

SCHEMBL14587739

CC(=O)c1ccc(-c2nc(NCc3ccc(C)cc3)c3ncn(C(C)C)c3n2)cc1

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 13/20 0.68
CDK5R1 Q15078 12/20 0.68
CDK1 P06493 6/20 0.68
CCNB2 O95067 5/20 0.68
CCNB1 P14635 5/20 0.68
CCNB3 Q8WWL7 5/20 0.68
CCNE2 O96020 4/20 0.55
CCNE1 P24864 4/20 0.55
CDK2 P24941 4/20 0.55
CCNA2 P20248 2/20 0.55
CCNA1 P78396 2/20 0.55
KDM4E B2RXH2 2/20 0.53
NPC1 O15118 2/20 0.53
MAPT P10636 2/20 0.53
TDP1 Q9NUW8 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5466623 0.90 CDK5 (0.78) CDK5CDK5R1CDK1CCNB2CCNB1
SCHEMBL14587744 0.88 CDK1 (0.64) CDK5CDK5R1CDK1CCNB2CCNB1
SCHEMBL21016776 0.77 CCNE2 (0.58) CDK5CDK5R1CDK1CCNB2CCNB1
SCHEMBL21016420 0.76 AHR (0.55) CDK5CDK5R1CDK1CCNB2CCNB1
SCHEMBL25261612 0.75 CCNK (0.55) CDK5CDK5R1CDK1CCNB2CCNB1
SCHEMBL30518531 0.75 CCNK (0.55) CDK5CDK5R1CDK1CCNB2CCNB1
SCHEMBL5466080 0.74 TDP1 (0.74) CDK5CDK5R1CDK1CCNB2CCNB1
SCHEMBL14431263 0.72 CDK1 (0.57) CDK5CDK5R1CDK1CCNB2CCNB1
SCHEMBL14587738 0.72 TDP1 (0.63) CDK5CDK5R1CDK1CCNB2CCNB1
SCHEMBL30518552 0.72 CCNK (0.60) CDK5CDK5R1CDK1CCNB2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176312-B2 Kinase inhibitor scaffolds and methods for their preparation THE SCRIPPS RESEARCH INSTITUTE (US) 2007-02-13 US disclosed