SCHEMBL14599488

SCHEMBL14599488

CCc1nn(CCO)c(C)c1Oc1cc(C#N)cc(C(N)=O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.40
PGR P06401 5/20 0.37
PARP15 Q460N3 1/20 0.33
PARP10 Q53GL7 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31
JAK3 P52333 1/20 0.31
F2 P00734 1/20 0.30
PRSS1 P07477 1/20 0.30
PRSS2 P07478 1/20 0.30
PRSS3 P35030 1/20 0.30
ST14 Q9Y5Y6 1/20 0.30
SLC2A1 P11166 1/20 0.30
SLC2A3 P11169 1/20 0.30
SLC2A4 P14672 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL509057 0.90 PGR (0.41) KCNH2PGRPARP15PARP10PARP2
SCHEMBL14599402 0.89 KCNH2 (0.49) KCNH2PGRALDH1A1LMNACYP3A4
SCHEMBL14620928 0.82 KCNH2 (0.43) KCNH2PGRALDH1A1LMNACYP3A4
Lersivirine SCHEMBL508446 0.78 KCNH2 (0.49) KCNH2PGRALDH1A1LMNACYP3A4
SCHEMBL5231006 0.78 KCNH2 (0.41) KCNH2PGRALDH1A1
SCHEMBL508505 0.78 PGR (0.40) KCNH2PGRPARP15PARP10PARP2
SCHEMBL2717137 0.77 KCNH2 (0.53) KCNH2PGRALDH1A1LMNACYP3A4
SCHEMBL14599354 0.76 KCNH2 (0.52) KCNH2PGR
Lersivirine SCHEMBL509058 0.76 KCNH2 (0.45) KCNH2PGRALDH1A1LMNA
SCHEMBL509168 0.75 KCNH2 (0.46) KCNH2PGRALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1762567-A1 Pyrazole derivatives for treating HIV Pfizer Limited (GB) 2007-03-14 EP disclosed