SCHEMBL14600768

SCHEMBL14600768

O=C(Nc1ccccc1)c1nc(-c2nncn2-c2cccc(F)c2F)c[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 3/20 0.36
GAA P10253 2/20 0.34
RIPK1 Q13546 2/20 0.34
DCLK1 O15075 1/20 0.34
DYRK3 O43781 1/20 0.34
ROCK2 O75116 1/20 0.34
PRKD3 O94806 1/20 0.34
MAP4K4 O95819 1/20 0.34
ABL1 P00519 1/20 0.34
EGFR P00533 1/20 0.34
NTRK1 P04629 1/20 0.34
LCK P06239 1/20 0.34
FYN P06241 1/20 0.34
CDK1 P06493 1/20 0.34
CSF1R P07333 1/20 0.34
LYN P07948 1/20 0.34
SRC P12931 1/20 0.34
MARK3 P27448 1/20 0.34
AXL P30530 1/20 0.34
FLT4 P35916 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14600767 0.82 GSK3B (0.36) GAARIPK1DCLK1DYRK3ROCK2
SCHEMBL5034026 0.80 MAPK7 (0.42) GAARIPK1DCLK1DYRK3ROCK2
SCHEMBL14600761 0.79 HPGD (0.42) MAP3K5LMNAPOLBALDH1A1KMT2A
SCHEMBL10067976 0.77 GSK3B (0.44) GAAGSK3BPOLBALDH1A1KMT2A
SCHEMBL5037204 0.70 NOTUM (0.36) DCLK1DYRK3ROCK2PRKD3MAP4K4
SCHEMBL14286143 0.67 MAPK1 (0.46) DCLK1DYRK3ROCK2PRKD3MAP4K4
SCHEMBL28063183 0.64 POLB (0.59) EGFRPOLBALDH1A1KMT2AMEN1
SCHEMBL23859765 0.63 FABP1 (0.48) LMNAPOLBATRALDH1A1KMT2A
SCHEMBL30075079 0.63 FABP1 (0.48) LMNAPOLBATRALDH1A1KMT2A
SCHEMBL14286148 0.63 MAPK1 (0.42) LMNAPOLBALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7169800-B2 Imidazole compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-01-30 US disclosed
US-7169800-B2 Imidazole compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-01-30 US disclosed