SCHEMBL14608968

SCHEMBL14608968

COc1ccnc2[nH]cc(C(O)c3ccc(N(Cc4ccc(C(F)(F)F)cc4)C(=O)OC(C)(C)C)nc3)c12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CETP P11597 4/20 0.32
LMNA P02545 1/20 0.32
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PDE2A O00408 3/20 0.31
CYP3A4 P08684 2/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
CCNT1 O60563 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CDK9 P50750 1/20 0.31
CCNA1 P78396 1/20 0.31
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31
GPR139 Q6DWJ6 1/20 0.31
CYP2C9 P11712 1/20 0.30
BRS3 P32247 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12927440 0.92 CETP (0.32) CETPLMNAALOX15TSHRHTT
SCHEMBL19302379 0.86 CYP3A4 (0.40) CETPLMNAALOX15TSHRHTT
SCHEMBL1267318 0.79 BRD4 (0.36) PDE2A
SCHEMBL641827 0.78 ACACB (0.30)
SCHEMBL858112 0.77 LMNA (0.39) LMNACYP3A4ROCK2CDK2CYP2C9
SCHEMBL1268055 0.74 RPS6KB1 (0.42)
SCHEMBL2112052 0.74 CYP3A4 (0.32) CYP3A4CYP2C9
SCHEMBL2114924 0.74 NTRK1 (0.32) CYP2C9
SCHEMBL3821880 0.74 CYP2C9 (0.42) SMN1; SMN2CYP3A4CYP2C9
SCHEMBL1266658 0.73 PDPK1 (0.36) ROCK2ROCK1CDK2CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007013896-A2 PYRROL (2,3-B) PYRIDINE DERIVATIVES PROTEIN KINASE INHIBITORS PLEXXIKON, INC. (US) 2007-02-01 WO disclosed