SCHEMBL14618844

SCHEMBL14618844

C=C(C)CN1CCC2(CC1)CN(C(=O)c1ccc(O)c(O)c1)c1ccccc12

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 6/20 0.50
HDAC6 Q9UBN7 6/20 0.50
NOTUM Q6P988 2/20 0.46
SLC18A3 Q16572 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
ALPL P05186 3/20 0.41
NSD2 O96028 1/20 0.41
GAA P10253 1/20 0.41
ALPG P10696 2/20 0.37
OPRD1 P41143 1/20 0.37
NPY5R Q15761 1/20 0.37
GPBAR1 Q8TDU6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5578816 0.85 HDAC1 (0.48) HDAC1HDAC6NOTUMGAA
SCHEMBL5578970 0.85 HDAC1 (0.49) HDAC1HDAC6NOTUMSLC18A3SIGMAR1
SCHEMBL5578576 0.83 HDAC1 (0.47) HDAC1HDAC6NOTUMSLC18A3SIGMAR1
SCHEMBL5578448 0.80 NOTUM (0.48) HDAC1HDAC6NOTUMSLC18A3SIGMAR1
SCHEMBL5578839 0.78 NOTUM (0.52) HDAC1HDAC6NOTUMSLC18A3SIGMAR1
SCHEMBL5579351 0.77 NOTUM (0.50) HDAC1HDAC6NOTUMSLC18A3SIGMAR1
SCHEMBL5578527 0.76 NOTUM (0.50) HDAC1HDAC6NOTUMSLC18A3SIGMAR1
SCHEMBL5578568 0.75 NOTUM (0.43) HDAC1HDAC6NOTUMSLC18A3SIGMAR1
SCHEMBL5578983 0.73 HDAC1 (0.53) HDAC1HDAC6NOTUMSLC18A3SIGMAR1
SCHEMBL14618521 0.73 HDAC1 (0.38) HDAC1HDAC6NOTUMSLC18A3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO disclosed