SCHEMBL14618521

SCHEMBL14618521

C=CCN1CCC2(CC1)CN(C(=O)c1ccc(O)c(O)c1)c1ccc(F)cc12

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
SIGMAR1 Q99720 2/20 0.37
SLC18A3 Q16572 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.35
ALDH1A1 P00352 2/20 0.34
GAA P10253 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
RECQL P46063 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
NSD2 O96028 1/20 0.33
ALPL P05186 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
NOTUM Q6P988 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5578712 0.91 HDAC1 (0.43) HDAC1HDAC6SIGMAR1SLC18A3PTGDR2
SCHEMBL5579054 0.88 CYP2D6 (0.44) HDAC1HDAC6ALDH1A1GAAHPGD
SCHEMBL5578500 0.87 HDAC1 (0.43) HDAC1HDAC6SIGMAR1SLC18A3NOTUM
SCHEMBL5578688 0.87 HDAC1 (0.48) HDAC1HDAC6SIGMAR1SLC18A3PTGDR2
SCHEMBL5578443 0.85 NOTUM (0.40) HDAC1HDAC6SIGMAR1SLC18A3PTGDR2
SCHEMBL5578784 0.85 TSHR (0.42) HDAC1HDAC6ALDH1A1GAAMAPT
SCHEMBL5578604 0.85 HDAC1 (0.36) HDAC1HDAC6SIGMAR1SLC18A3PTGDR2
SCHEMBL5578768 0.85 HDAC1 (0.41) HDAC1HDAC6ALDH1A1KDM4ELMNA
SCHEMBL5578902 0.85 NQO2 (0.41) HDAC1HDAC6PTGDR2ALDH1A1
SCHEMBL14618893 0.85 OPRM1 (0.43) HDAC1HDAC6SIGMAR1SLC18A3OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO disclosed