SCHEMBL1462017

SCHEMBL1462017

C=C(C)c1nc(C2CCCOCC2)cc(C)c1[N+](=O)[O-]

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.34
MAPK1 P28482 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
ALDH1A1 P00352 6/20 0.32
MAPT P10636 2/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
KDM5B Q9UGL1 1/20 0.31
GAA P10253 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1461741 0.73 ALDH1A1 (0.48) KMT2AMAPK1NPSR1ALDH1A1MAPT
SCHEMBL1461584 0.69 ALDH1A1 (0.34) KMT2AMAPK1NPSR1ALDH1A1MAPT
SCHEMBL21543246 0.67 POLB (0.37) KMT2AALDH1A1MAPTCYP1A2TDP1
SCHEMBL27227005 0.61 MAPT (0.41) ALDH1A1MAPTCYP1A2CYP2C9GAA
SCHEMBL31020485 0.60 ALDH1A1 (0.44) KMT2AALDH1A1MAPTTDP1
SCHEMBL29427889 0.60 MAPT (0.43) KMT2AMAPK1ALDH1A1MAPTTDP1
SCHEMBL28929673 0.60 MAPT (0.43) KMT2AMAPK1ALDH1A1MAPTTDP1
SCHEMBL27365047 0.59 ALDH1A1 (0.42) KMT2AALDH1A1MAPTCYP1A2CYP2C9
SCHEMBL20516345 0.58 ALDH1A1 (0.34) KMT2AALDH1A1MAPTCYP1A2CYP2C9
SCHEMBL14183096 0.58 GAA (0.50) KMT2AMAPK1ALDH1A1MAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011026891-A1 SUBSTITUTED PYRIDINE DERIVATIVES AND THEIR MEDICAL USE NEUROSEARCH A/S (DK) 2011-03-10 WO disclosed