SCHEMBL14624005

SCHEMBL14624005

CS(=O)(=O)c1cccc(-c2ccc(-c3cc(C(F)(F)F)nn3-c3cccc(OC(N)=O)c3)s2)c1

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RXRA P19793 7/20 0.61
NR1H2 P55055 7/20 0.61
NR1H3 Q13133 7/20 0.61
PTGS2 P35354 6/20 0.47
KLKB1 P03952 1/20 0.44
PTGS1 P23219 2/20 0.43
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3471811 0.90 RXRA (0.65) RXRANR1H2NR1H3PTGS2PTGS1
SCHEMBL3471365 0.90 RXRA (0.60) RXRANR1H2NR1H3PTGS2KLKB1
SCHEMBL3471279 0.90 RXRA (0.60) RXRANR1H2NR1H3PTGS2KLKB1
SCHEMBL3471406 0.88 RXRA (0.67) RXRANR1H2NR1H3PTGS2PTGS1
SCHEMBL3475519 0.87 RXRA (0.57) RXRANR1H2NR1H3PTGS2KLKB1
SCHEMBL3473874 0.86 NR1H2 (0.67) RXRANR1H2NR1H3PTGS2PTGS1
SCHEMBL3471400 0.86 RXRA (0.60) RXRANR1H2NR1H3PTGS2KLKB1
SCHEMBL3473141 0.86 RXRA (0.60) RXRANR1H2NR1H3PTGS2KLKB1
SCHEMBL3471667 0.86 RXRA (0.56) RXRANR1H2NR1H3PTGS2KLKB1
SCHEMBL3472855 0.85 RXRA (0.64) RXRANR1H2NR1H3PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007002559-A1 PYRAZOLE BASED LXR MODULATORS EXELIXIS, INC. (US) 2007-01-04 WO disclosed