SCHEMBL14625499

SCHEMBL14625499

COC(=O)C(C(=O)OC)[C@@H](NC=O)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.58
TSHR P16473 2/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
MEN1 O00255 2/20 0.41
ALDH1A1 P00352 2/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
LMNA P02545 1/20 0.41
TACR1 P25103 1/20 0.39
CYP2D6 P10635 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
KLK7 P49862 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28192047 0.85 KMT2A (0.56) KMT2ATSHRCYP3A4CYP2C19MEN1
SCHEMBL206552 0.80 KMT2A (0.49) KMT2ATSHRMEN1ALDH1A1LMNA
SCHEMBL11991382 0.79 KMT2A (0.61) KMT2ATSHRCYP3A4MEN1ALDH1A1
SCHEMBL8505416 0.79 KMT2A (0.61) KMT2ATSHRCYP3A4MEN1ALDH1A1
SCHEMBL14624894 0.78 CYP3A4 (0.55) KMT2ATSHRCYP3A4CYP2C19MEN1
SCHEMBL13024506 0.78 KMT2A (0.55) KMT2ACYP3A4CYP2C19MEN1ALDH1A1
SCHEMBL12789448 0.74 KMT2A (0.48) KMT2AMEN1ALDH1A1TACR1CYP2D6
SCHEMBL7415448 0.74 KMT2A (0.43) KMT2ATSHRCYP3A4CYP2C19MEN1
SCHEMBL7818496 0.73 KMT2A (0.41) KMT2ATSHRCYP2C19MEN1ALDH1A1
SCHEMBL24576212 0.73 KMT2A (0.43) KMT2ATSHRCYP3A4CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007011910-A2 CHIRAL AMINE-CATALYZED ASYMMETRIC ADDITION OF CARBON-CENTERED NUCLEOPHILES TO IMINES TRUSTEES OF BOSTON UNIVERSITY (US) 2007-01-25 WO disclosed