SCHEMBL14629964

SCHEMBL14629964

C#Cc1nc(C(F)(F)F)ccc1N

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
KDM4E B2RXH2 6/20 0.32
HSD17B10 Q99714 2/20 0.32
ALDH1A1 P00352 4/20 0.32
TRPV4 Q9HBA0 1/20 0.31
MAT2A P31153 1/20 0.31
P2RX7 Q99572 1/20 0.31
KMT2A Q03164 1/20 0.31
CA2 P00918 1/20 0.31
CHKA P35790 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30032746 0.81 ALDH1A1 (0.36) HSP90AA1HSP90AB1KDM4EHSD17B10ALDH1A1
SCHEMBL2159069 0.81 ALDH1A1 (0.36) HSP90AA1HSP90AB1KDM4EHSD17B10ALDH1A1
SCHEMBL14630424 0.75 HSP90AA1 (0.36) HSP90AA1HSP90AB1KDM4EALDH1A1PTGS2
SCHEMBL898882 0.73 HSP90AA1 (0.38) HSP90AA1HSP90AB1KDM4EHSD17B10ALDH1A1
SCHEMBL29745069 0.73 HSP90AA1 (0.38) HSP90AA1HSP90AB1KDM4EHSD17B10ALDH1A1
SCHEMBL25371113 0.71 HSP90AA1 (0.36) HSP90AA1HSP90AB1KDM4EHSD17B10ALDH1A1
Hydrochloric Acid SCHEMBL14127591 0.71 HSP90AA1 (0.36) HSP90AA1HSP90AB1KDM4EHSD17B10ALDH1A1
SCHEMBL830696 0.71 HSP90AA1 (0.36) HSP90AA1HSP90AB1KDM4EHSD17B10ALDH1A1
SCHEMBL30303053 0.71 HSP90AA1 (0.36) HSP90AA1HSP90AB1KDM4EHSD17B10ALDH1A1
SCHEMBL24169965 0.70 PDPK1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013010880-A1 NEW CRTH2 ANTAGONISTS ALMIRALL, S.A. (ES) 2013-01-24 WO disclosed
EP-2548876-A1 New CRTh2 antagonists Almirall, S.A. (ES) 2013-01-23 EP disclosed