SCHEMBL14630965

SCHEMBL14630965

O=C1CCN(C(=O)OCc2ccccc2)C(Cc2ccccc2)C1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 2/20 0.53
PSEN2 P49810 2/20 0.53
APH1B Q8WW43 2/20 0.53
NCSTN Q92542 2/20 0.53
APH1A Q96BI3 2/20 0.53
PSENEN Q9NZ42 2/20 0.53
PARP1 P09874 1/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
CYP2C19 P33261 2/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
ELANE P08246 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21326064 0.89 PARP1 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL21751143 0.89 PARP1 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL19389930 0.88 PARP1 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8726172 0.85 RAB9A (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1660359 0.85 ELANE (0.55) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL754805 0.84 HTR2C (0.54) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1170552 0.84 HTR2C (0.54) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL31329634 0.84 HTR2C (0.54) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2088860 0.84 ABCB1 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL15352939 0.84 ABCB1 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2548877-A1 4-(5-Membered fused pyridinyl)benzamides as BTK-inhibitors MSD Oss B.V. (NL) 2013-01-23 EP disclosed