SCHEMBL14632161

SCHEMBL14632161

CCOC(=O)OC1=C(C)N(c2cccc(C(F)(F)F)c2)c2nnnn2C1c1ccc(C#N)cc1

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ELANE P08246 20/20 0.59
CYP3A4 P08684 4/20 0.54
CYP2C9 P11712 6/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14632050 1.00 ELANE (0.59) ELANECYP3A4CYP2C9
SCHEMBL14632068 0.91 ELANE (0.54) ELANECYP3A4CYP2C9
SCHEMBL230899 0.88 ELANE (0.72) ELANECYP3A4CYP2C9
SCHEMBL230520 0.88 ELANE (0.72) ELANECYP3A4CYP2C9
SCHEMBL1746677 0.87 ELANE (0.58) ELANECYP3A4CYP2C9
SCHEMBL232930 0.84 ELANE (0.62) ELANECYP3A4CYP2C9
SCHEMBL14632007 0.84 ELANE (0.55) ELANECYP3A4CYP2C9
SCHEMBL231686 0.84 ELANE (0.57) ELANECYP3A4CYP2C9
SCHEMBL15456300 0.84 ELANE (0.57) ELANECYP3A4CYP2C9
SCHEMBL14632131 0.83 ELANE (0.54) ELANECYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2385945-B1 TRIAZOLO AND TETRAZOLO PYRIMIDINE DERIVATIVES AS HNE INHIBITORS FOR TREATING COPD BAYER IP GMBH (DE) 2013-01-23 EP disclosed