SCHEMBL14637784

SCHEMBL14637784

CC1(NC(=O)O)CCCN(c2ccc(C(F)(F)F)cc2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.44
FPR1 P21462 1/20 0.43
FPR2 P25090 1/20 0.43
NOTUM Q6P988 1/20 0.43
USP2 O75604 4/20 0.43
HIF1A Q16665 4/20 0.43
CYP2C9 P11712 3/20 0.43
TSHR P16473 2/20 0.43
CYP2D6 P10635 1/20 0.43
PTGES O14684 2/20 0.42
CA12 O43570 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
SLC6A9 P48067 3/20 0.41
AKR1C3 P42330 1/20 0.40
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15106363 0.81 FPR2 (0.44) CYP3A4FPR1FPR2NOTUMUSP2
SCHEMBL15106364 0.81 FPR2 (0.44) CYP3A4FPR1FPR2NOTUMUSP2
SCHEMBL15115344 0.80 CYP3A4 (0.44) CYP3A4FPR1FPR2NOTUMUSP2
SCHEMBL23387362 0.75 CYP11B1 (0.43) CYP3A4HIF1ATSHR
SCHEMBL23387360 0.75 CYP11B1 (0.43) CYP3A4HIF1ATSHR
SCHEMBL14637697 0.74 CYP3A4 (0.40) CYP3A4FPR1FPR2NOTUMUSP2
SCHEMBL14638114 0.74 CYP3A4 (0.40) CYP3A4FPR1FPR2NOTUMUSP2
SCHEMBL14650106 0.73 FPR2 (0.38) CYP3A4FPR1FPR2NOTUMUSP2
SCHEMBL15106532 0.73 FPR2 (0.38) CYP3A4FPR1FPR2NOTUMUSP2
SCHEMBL15106531 0.73 FPR2 (0.38) CYP3A4FPR1FPR2NOTUMUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8815909-B2 Diaminocyclohexane compounds and uses thereof BRISTOL-MYERS SQUIBB COMPANY (US) 2014-08-26 US disclosed
US-20130184284-A1 DIAMINOCYCLOHEXANE COMPOUNDS AND USES THEREOF BRISTOL-MYERS SQUIBB COMPANY 2013-07-18 US disclosed
WO-2013012827-A1 DIAMINOCYCLOHEXANE COMPOUNDS AND USES THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 2013-01-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130184284-A1 DIAMINOCYCLOHEXANE COMPOUNDS AND USES THEREOF NPY4R, NPY2R, NPY1R CYP3A4 1357/4885FPR1 28/4885FPR2 39/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.