SCHEMBL14641817

SCHEMBL14641817

CC(C)N(C)Cc1ccc(C(F)(F)F)nc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.42
KCNH2 Q12809 3/20 0.41
DAO P14920 3/20 0.39
TKT P29401 1/20 0.38
KDM1A O60341 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
CYP2C8 P10632 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
TRPV3 Q8NET8 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14540447 0.78 KCNH2 (0.45) KCNH2DAOLMNACYP2C8CYP2D6
SCHEMBL8171813 0.76 TRPV4 (0.47) TRPV4DAOTKTKDM1AMAOA
SCHEMBL14641819 0.75 SMN1; SMN2 (0.44) KDM4ELMNAGAASMN1; SMN2
SCHEMBL4237439 0.73 TRPV4 (0.44) TRPV4DAOTKTKDM1AMAOA
SCHEMBL3819747 0.73 HTR2A (0.47) TRPV4MAOA
SCHEMBL12197882 0.73 DAO (0.47) TRPV4DAOTKTKDM1AMAOA
SCHEMBL91511 0.73 TRPV4 (0.52) TRPV4KCNH2DAOTKTKDM1A
SCHEMBL24973120 0.72 TRPV4 (0.43) TRPV4DAOTKTKDM1AMAOA
SCHEMBL19764842 0.72 TRPV4 (0.43) TRPV4DAOTKTKDM1AMAOA
SCHEMBL12844982 0.72 KDM1A (0.47) TRPV4KDM1AMAOAMAOBCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8354414-B2 Substituted bicyclic pyrimidines CEPHALON, INC (US) 2013-01-15 US disclosed