SCHEMBL14645

SCHEMBL14645

O[C@]12CCCCC1COC[C@H]2Nc1ccc(F)c(F)c1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 10/20 0.53
TRPC5 Q9UL62 2/20 0.42
HRH2 P25021 1/20 0.42
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SLC6A3 Q01959 2/20 0.39
ESR1 P03372 1/20 0.39
PGR P06401 1/20 0.39
HTR2A P28223 1/20 0.39
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
BACE1 P56817 2/20 0.34
BACE2 Q9Y5Z0 2/20 0.34
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11954725 1.00 TRPA1 (0.53) TRPA1TRPC5HRH2NPC1RAB9A
SCHEMBL11966017 1.00 TRPA1 (0.53) TRPA1TRPC5HRH2NPC1RAB9A
SCHEMBL15809914 1.00 TRPA1 (0.53) TRPA1TRPC5HRH2NPC1RAB9A
SCHEMBL11967515 0.86 TRPA1 (0.71) TRPA1TRPC5HRH2NPC1RAB9A
SCHEMBL11971240 0.86 TRPA1 (0.71) TRPA1TRPC5HRH2NPC1RAB9A
SCHEMBL11227 0.86 TRPA1 (0.71) TRPA1TRPC5HRH2NPC1RAB9A
SCHEMBL3120 0.86 TRPA1 (0.71) TRPA1TRPC5HRH2NPC1RAB9A
SCHEMBL11895423 0.85 TRPA1 (0.73) TRPA1TRPC5HRH2NPC1RAB9A
SCHEMBL15809851 0.84 TRPA1 (0.52) TRPA1TRPC5HRH2NPC1RAB9A
SCHEMBL2522 0.84 TRPA1 (0.52) TRPA1TRPC5HRH2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011043954-A1 NOVEL TRPA1 ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-04-14 WO disclosed