SCHEMBL14646451

SCHEMBL14646451

CCOP(=O)(O)Cc1cc2cccnc2s1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.51
AKR1B1 P15121 1/20 0.39
MET P08581 1/20 0.36
CHRNA7 P36544 1/20 0.34
KDM4E B2RXH2 2/20 0.34
MAPT P10636 2/20 0.34
RXFP1 Q9HBX9 2/20 0.34
MAPK1 P28482 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP2C9 P11712 2/20 0.34
THRB P10828 1/20 0.34
CASP1 P29466 1/20 0.34
RAD52 P43351 1/20 0.34
CASP7 P55210 1/20 0.34
CASP6 P55212 1/20 0.34
CASP8 Q14790 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10245795 0.88 CYP2A6 (0.52) CYP2A6AKR1B1METCHRNA7KDM4E
SCHEMBL7021081 0.75 CYP2A6 (0.68) CYP2A6AKR1B1METMAPTALDH1A1
SCHEMBL6978499 0.72 RAB9A (0.43) KDM4EALDH1A1CASP6SMN1; SMN2NPC1
SCHEMBL2175943 0.72 CYP2A6 (0.63) CYP2A6AKR1B1METCHRNA7KDM4E
Methylethylamine SCHEMBL25352737 0.69 CYP2A6 (0.72) CYP2A6AKR1B1METKDM4EMAPT
SCHEMBL10469274 0.69 CYP2A6 (0.59) CYP2A6AKR1B1METMAPTNPC1
SCHEMBL10423641 0.69 CYP2A6 (0.63) CYP2A6AKR1B1METKDM4EMAPT
SCHEMBL2174717 0.69 CYP2A6 (0.63) CYP2A6AKR1B1METKDM4EMAPT
SCHEMBL31207840 0.69 KDM4E (0.48) CYP2A6CHRNA7KDM4EMAPTNPSR1
SCHEMBL10245531 0.69 KDM4E (0.48) CYP2A6CHRNA7KDM4EMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029614-B1 COLD MENTHOL RECEPTOR-1 ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2013-01-23 EP disclosed