SCHEMBL14647899

SCHEMBL14647899

O=C(c1ccc2c(ccn2-c2cc(F)cc(F)c2)c1)N1CC(N2CCN(C(=O)c3nccs3)CC2)C1

nearest known ligand 0.87

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 20/20 0.87
FAAH O00519 1/20 0.87

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL698521 0.93 MGLL (1.00) MGLLFAAH
SCHEMBL14647981 0.92 MGLL (0.83) MGLLFAAH
SCHEMBL697821 0.90 MGLL (0.85) MGLLFAAH
SCHEMBL14647893 0.90 MGLL (0.84) MGLLFAAH
SCHEMBL911461 0.89 MGLL (0.81) MGLLFAAH
SCHEMBL911357 0.88 MGLL (0.85) MGLLFAAH
SCHEMBL910669 0.88 MGLL (0.85) MGLLFAAH
SCHEMBL912325 0.88 MGLL (0.84) MGLLFAAH
SCHEMBL14827113 0.88 MGLL (0.84) MGLLFAAH
SCHEMBL14647931 0.88 MGLL (0.79) MGLLFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421823-B1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2015-01-14 EP disclosed
EP-2421825-B9 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2014-08-20 EP disclosed
EP-2421825-B1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2014-01-01 EP disclosed
US-8362000-B2 Azetidinyl diamides as monoacylglycerol lipase inhibitors JANSSEN PHARMACEUTICA NV (BE) 2013-01-29 US disclosed