SCHEMBL14654247

SCHEMBL14654247

O=C(OCc1ccccc1)N1CCCC(c2ncc3c(Cl)nccn23)C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.47
JAK1 P23458 3/20 0.47
TYK2 P29597 2/20 0.47
JAK3 P52333 2/20 0.47
LCK P06239 2/20 0.43
GRIN2B Q13224 5/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
CYP2D6 P10635 3/20 0.42
CYP2C9 P11712 3/20 0.42
CYP3A4 P08684 2/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
CYP2C19 P33261 1/20 0.41
MAPK1 P28482 1/20 0.41
USP30 Q70CQ3 1/20 0.41
BCL9 O00512 2/20 0.40
CTNNB1 P35222 2/20 0.40
IGF1R P08069 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14647469 1.00 JAK2 (0.47) JAK2JAK1TYK2JAK3LCK
SCHEMBL28938318 0.95 SMN1; SMN2 (0.46) JAK2JAK1TYK2JAK3GRIN2B
SCHEMBL21050978 0.95 SMN1; SMN2 (0.46) JAK2JAK1TYK2JAK3GRIN2B
SCHEMBL2323323 0.91 OPRD1 (0.43) JAK2JAK1TYK2JAK3GRIN2B
SCHEMBL593236 0.90 SMN1; SMN2 (0.50) JAK2JAK1TYK2JAK3GRIN2B
SCHEMBL30449894 0.88 KMT2A (0.40) JAK2JAK1TYK2JAK3LCK
SCHEMBL2323403 0.85 GRIN2B (0.43) GRIN2BSMN1; SMN2NPC1RAB9ACYP2D6
SCHEMBL2323399 0.85 GRIN2B (0.43) GRIN2BSMN1; SMN2NPC1RAB9ACYP2D6
SCHEMBL14651431 0.84 BTK (0.47)
SCHEMBL15762428 0.84 BTK (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013010380-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-01-24 WO disclosed