SCHEMBL14664468

SCHEMBL14664468

CC(=O)[C@@H]1C[C@@H]2C[C@@H]2N1C(=O)[C@@H](NC(=O)OC(C)(C)C)C12CC3CC(CC(O)(C3)C1)C2

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 15/20 0.42
DPP8 Q6V1X1 2/20 0.42
DPP9 Q86TI2 2/20 0.42
CYP3A4 P08684 1/20 0.42
HSD11B1 P28845 1/20 0.32
ITGB3 P05106 1/20 0.31
ITGA2B P08514 1/20 0.31
MEN1 O00255 1/20 0.31
MAPK1 P28482 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14410140 1.00 DPP4 (0.42) DPP4DPP8DPP9CYP3A4HSD11B1
SCHEMBL14554067 0.91 DPP4 (0.43) DPP4DPP8DPP9CYP3A4
SCHEMBL2434106 0.91 DPP4 (0.43) DPP4DPP8DPP9CYP3A4
SCHEMBL8269749 0.91 DPP4 (0.43) DPP4DPP8DPP9CYP3A4
SCHEMBL8277771 0.91 DPP4 (0.43) DPP4DPP8DPP9CYP3A4
SCHEMBL8276954 0.91 DPP4 (0.43) DPP4DPP8DPP9CYP3A4
SCHEMBL15149979 0.91 DPP4 (0.43) DPP4DPP8DPP9CYP3A4
SCHEMBL12969791 0.88 DPP4 (0.43) DPP4DPP8DPP9CYP3A4HSD11B1
SCHEMBL8271030 0.85 DPP4 (0.62) DPP4DPP8DPP9CYP3A4
SCHEMBL13404730 0.85 DPP4 (0.41) DPP4DPP8DPP9CYP3A4HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8361761-B2 Process for preparing dipeptidyl peptidase IV inhibitors and intermediates therefor BRISTOL MYERS-SQUIBB COMPANY (US) 2013-01-29 US disclosed