SCHEMBL14670320

SCHEMBL14670320

Cc1cc(Nc2ccn[nH]2)nc(N2CCC[C@@H](NC(=O)O)C2)n1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.48
TSHR P16473 3/20 0.48
GAA P10253 2/20 0.48
KDM4E B2RXH2 6/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
KMT2A Q03164 1/20 0.46
RET P07949 2/20 0.45
CCNE1 P24864 3/20 0.42
CDK2 P24941 3/20 0.42
ROCK2 O75116 3/20 0.42
ROCK1 Q13464 2/20 0.42
POLB P06746 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14670299 1.00 HSD17B10 (0.48) HSD17B10TSHRGAAKDM4EMEN1
SCHEMBL473587 0.87 KDM4E (0.64) HSD17B10TSHRGAAKDM4EMEN1
Trifluoroacetic Acid SCHEMBL342591 0.83 KDM4E (0.57) HSD17B10TSHRGAAKDM4EMEN1
Trifluoroacetic Acid SCHEMBL341448 0.83 KDM4E (0.57) HSD17B10TSHRGAAKDM4EMEN1
SCHEMBL342269 0.82 KDM4E (0.41) HSD17B10TSHRGAAKDM4EMEN1
SCHEMBL342930 0.82 KDM4E (0.41) HSD17B10TSHRGAAKDM4EMEN1
Trifluoroacetic Acid SCHEMBL342230 0.81 NAPEPLD (0.42) HSD17B10GAAKDM4EMEN1ALDH1A1
SCHEMBL341449 0.79 KDM4E (0.45) HSD17B10TSHRGAAKDM4EMEN1
SCHEMBL342592 0.79 KDM4E (0.45) HSD17B10TSHRGAAKDM4EMEN1
SCHEMBL3812064 0.78 RET (0.60) HSD17B10TSHRGAARETCCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367690-B2 Aminopyridine derivatives having aurora a selective inhibitory action VERTEX PHARMACEUTICALS INC. (US) 2013-02-05 US disclosed