SCHEMBL14679151

SCHEMBL14679151

Cc1ccc(NC(=O)CCNC(=O)OC(C)(C)C)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.60
CA2 P00918 2/20 0.60
POLB P06746 4/20 0.53
HDAC8 Q9BY41 3/20 0.50
HDAC3 O15379 2/20 0.50
HDAC1 Q13547 2/20 0.50
HDAC2 Q92769 2/20 0.50
HDAC10 Q969S8 2/20 0.50
HDAC11 Q96DB2 2/20 0.50
HDAC6 Q9UBN7 2/20 0.50
HDAC4 P56524 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC9 Q9UKV0 1/20 0.50
HDAC5 Q9UQL6 1/20 0.50
NCOR2 Q9Y618 1/20 0.49
KMT2A Q03164 2/20 0.48
NPC1 O15118 1/20 0.48
TP53 P04637 1/20 0.48
RAB9A P51151 1/20 0.48
CCNC P24863 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8692897 0.94 CA1 (0.66) CA1CA2POLBHDAC8HDAC3
SCHEMBL4757472 0.87 CA1 (0.59) CA1CA2POLBKMT2ANPC1
SCHEMBL937131 0.87 CA1 (0.59) CA1CA2POLBHDAC8HDAC3
SCHEMBL6274441 0.87 CA1 (0.58) CA1CA2HDAC8HDAC3HDAC1
SCHEMBL3955534 0.86 CA1 (0.65) CA1CA2POLBHDAC8HDAC3
SCHEMBL14679376 0.85 POLB (0.54) CA1CA2POLBHDAC8HDAC3
SCHEMBL4758298 0.85 CA1 (0.57) CA1CA2POLBHDAC8HDAC3
SCHEMBL4412010 0.85 CA1 (0.57) CA1CA2HDAC8HDAC3HDAC1
SCHEMBL4625768 0.85 MAPT (0.57) CA1CA2POLBHDAC8HDAC3
SCHEMBL14679432 0.84 CA1 (0.60) CA1CA2POLBHDAC8HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367668-B2 Pyridazinone derivatives MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 2013-02-05 US disclosed
US-8367668-B2 Pyridazinone derivatives MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 2013-02-05 US disclosed