SCHEMBL14686151

SCHEMBL14686151

COc1ccc(Cc2c(N)nn3ccnc3c2N)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
CYP2D6 P10635 1/20 0.49
ATM Q13315 1/20 0.49
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.40
POLB P06746 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
HPGD P15428 1/20 0.38
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
HSP90AB1 P08238 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
LTA4H P09960 2/20 0.36
PDE2A O00408 1/20 0.35
CSF1R P07333 1/20 0.35
PI4KA P42356 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28604914 0.77 ALDH1A1 (0.49) ALDH1A1CYP2D6ATMLMNASMN1; SMN2
Hydrochloric Acid SCHEMBL7522555 0.71 ALDH1A1 (0.68) ALDH1A1CYP2D6ATMLMNASMN1; SMN2
SCHEMBL28729752 0.71 ALDH1A1 (0.58) ALDH1A1CYP2D6ATMLMNASMN1; SMN2
SCHEMBL29433996 0.71 ALDH1A1 (0.58) ALDH1A1CYP2D6ATMLMNASMN1; SMN2
SCHEMBL8097615 0.70 ALDH1A1 (0.65) ALDH1A1CYP2D6ATMLMNASMN1; SMN2
SCHEMBL28996034 0.70 ALDH1A1 (0.56) ALDH1A1CYP2D6ATMLMNASMN1; SMN2
SCHEMBL29687392 0.70 ALDH1A1 (0.56) ALDH1A1CYP2D6ATMLMNASMN1; SMN2
SCHEMBL28054249 0.69 ALDH1A1 (0.59) ALDH1A1CYP2D6ATMLMNASMN1; SMN2
SCHEMBL23045757 0.68 ALDH1A1 (0.58) ALDH1A1CYP2D6ATMLMNASMN1; SMN2
SCHEMBL13841864 0.68 MAOB (0.56) CYP2D6LTA4HPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928879-B1 FUSED HETEROCYCLIC COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL MYERS SQUIBB CO (US) 2013-02-13 EP claimed